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Obstacles and innovations of macrocyclic drug development

Drug Target Review

3 Antibodies are primarily used to target extracellular proteins, though researchers have generated antibodies that can reach intracellular targets. Metabolism was another concern in the early development of macrocyclic peptides. Ajay N Jain Ajay is VP of Research for the Optibrium s BioPharmics Division. Springer, 2019.